A New and Simple Synthesis of Sulfonyl Ureas from Sulfonamides and N-Alkyl-1,2,4-dithiazolidine-3,5-diones. R.K. Gessner and K. Chibale*. Synlett. 2009, 17, 2839-2843.


Pharmacologically relevant bifunctional compounds containing chloroquinoline and dihydropyrimidone moieties; syntheses and crystal structures of a target molecule and selected intermediates. N. D. Watermeyer, K. Chibale* and M.R. Caira*. J. Chem. Crystallography. 2009, 39, (10), 753-760.


Cycloaddition and One-Carbon Homologation Studies in the Synthesis of Advanced Iridoid Precursors. A. T. Stevens, M. R. Caira, J. R. Bull, and K. Chibale* Org. Biomol. Chem., 2009, 7, 3527- 3536.


Synthesis of novel anti-2-alkoxy-3-amino-3-arylpropan-1-ols and cis-5-alkoxy-4aryl-1,3-oxazinanes with antimalarial activity. M. D’hooghe, P. J. Smith, S. Dekeukeleire, K. Mollet, K. Chibale and N. De Kimpe* J. Med. Chem. 2009, 52, 4058-4062.


Novel web-based tools combining chemistry informatics, biology and social networks for drug discovery. M. Hohman, K. Gregory, K. Chibale, P.J. Smith, S. Ekins and B. Bunin*. Drug Discovery Today, 2009,14, 261-70.


Synthetic Medicinal Chemistry of Antimalarial Natural Products. V. Kumar, A. Mahajan, and K. Chibale*. Bioorg. Med. Chem. 2009, 17, 2236-2275. Paper ranked in the top ten of the most popular/most-cited articles for 2009 - 2010 academic year in this journal.